Vardenafil hydrochloride trihydrate
CAS No. 330808-88-3
Vardenafil hydrochloride trihydrate ( BAY 38-9456;Vardenafil HCl; Levitra; Staxyn; Vivanza )
Catalog No. M18429 CAS No. 330808-88-3
Vardenafil HCl Trihydrate is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 35 | Get Quote |
|
10MG | 58 | Get Quote |
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25MG | 114 | Get Quote |
|
50MG | 177 | Get Quote |
|
100MG | 282 | Get Quote |
|
200MG | 421 | Get Quote |
|
500MG | 678 | Get Quote |
|
1G | Get Quote | Get Quote |
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Biological Information
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Product NameVardenafil hydrochloride trihydrate
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NoteResearch use only, not for human use.
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Brief DescriptionVardenafil HCl Trihydrate is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.
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DescriptionVardenafil, also known as BAY 38-9456, is a PDE5 inhibitor used for treating erectile dysfunction. Vardenafil (VAR) is synthetic, highly selective, and potent inhibitor of phosphodiesterase-5 which competitively inhibits cyclic guanosine monophosphate (cGMP) hydrolysis and thus increases cGMP levels. It is clinically approved for treatment of erectile dysfunction in men, including diabetic and postprostatectomy patients.
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SynonymsBAY 38-9456;Vardenafil HCl; Levitra; Staxyn; Vivanza
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PathwayOthers
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TargetOther Targets
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RecptorPDE1; PDE5
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number330808-88-3
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Formula Weight579.11
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Molecular FormulaC23H32N6O4S·HCl·3H2O
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Purity98%
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Solubility——
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SMILESn12[nH]c(nc(=O)c1c(nc2CCC)C)c1c(ccc(c1)S(=O)(=O)N1CCN(CC1)CC)OCC.Cl.O.O.O
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Chemical Name2-(2-ethoxy-5-((4-ethylpiperazin-1-yl)sulfonyl)phenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(1H)-one dihydrochloride trihydrate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1 Saenz de Tejada I, et al. Int J Impot Res, 2001, 13(5), 282-290.
molnova catalog
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